The cysteinyl leukotriene receptors (CysLTRs) include the following two receptors:
The recently elucidated CysLTE, represented by GPR99/OXGR1, may constitute a third CysLTR.[1]
See also
References
|  | 
|---|
| Receptor (ligands)
 | | BLTTooltip Leukotriene B4 receptor | | BLT1Tooltip Leukotriene B4 receptor 1 | 
Antagonists: 20-Carboxy-LTB4AmelubantCGS-23131 (LY-223982)CGS-25019CCP-105696CP-195543EtalocibLY-293111MoxilubantONO-4057RG-14893RP-69698SB-209247SC-53228TicolubantU-75302ZK-158252
 | 
|---|
 | BLT2Tooltip Leukotriene B4 receptor 2 | 
Antagonists: CP-195543LY-255283ZK-158252
 | 
|---|
 | 
|---|
 | Tooltip Cysteinyl leukotriene receptor | | CysLT1Tooltip Cysteinyl leukotriene receptor 1 | 
Antagonists: AblukastBAYu9773BAYu9916BAYx7195CinalukastFPL-55712ICI-198615IralukastLY-170680MasilukastMK-571MontelukastONO-1078PobilukastPranlukastRitolukastSKF-104353SR-2640SulukastTipelukastTomelukastVerlukastZafirlukastZD-3523
 | 
|---|
 | CysLT2Tooltip Cysteinyl leukotriene receptor 2 | 
Antagonists: BAYu9773BAYu9916
 | 
|---|
 | CysLTETooltip Cysteinyl leukotriene receptor E |  | 
|---|
 | 
|---|
 | 
|---|
| Enzyme (inhibitors)
 | | 5-LOXTooltip Arachidonate 5-lipoxygenase | 
FLAPTooltip Arachidonate 5-lipoxygenase-activating protein inhibitors: AM-103AM-679BAYx1005MK-591MK-886
 | 
|---|
 | 12-LOXTooltip Arachidonate 12-lipoxygenase |  | 
|---|
 | 15-LOXTooltip Arachidonate 15-lipoxygenase |  | 
|---|
 | LTA4HTooltip Leukotriene A4 hydrolase |  | 
|---|
 | LTB4HTooltip Leukotriene B4 ω-hydroxylase |  | 
|---|
 | LTC4STooltip Leukotriene C4 synthase |  | 
|---|
 | LTC4HTooltip Leukotriene C4 hydrolase |  | 
|---|
 | LTD4Tooltip Leukotriene D4 hydrolase |  | 
|---|
 | 
|---|
| Others |  | 
|---|
| 
See alsoReceptor/signaling modulatorsProstanoid signaling modulators
 |